PPARgamma LBD complexed with MRL24
GQLNPESADL RALAKHLYDS YIKSFPLTKA KARAILTGKT TDKSPFVIYD MNSLMMGEDK IKFKHITPLQ EQSKEVAIRI FQGCQFRSVE AVQEITEYAK SIPGFVNLDL NDQVTLLKYG VHEIIYTMLA SLMNKDGVLI SEGQGFMTRE FLKSLRKPFG DFMEPKFEFA VKFNALELDD SDLAIFIAVI ILSGDRPGLL NVKPIEDIQD NLLQALELQL KLNHPESSQL FAKLLQKMTD LRQIVTEHVQ LLQVIKKTET DMSLHPLLQE IYKDLY
Polymer type: polypeptide(L)
Total | 1H | 13C | 15N | |
---|---|---|---|---|
All | 33.3 % (1120 of 3368) | 18.8 % (331 of 1757) | 45.0 % (594 of 1320) | 67.0 % (195 of 291) |
Backbone | 58.9 % (962 of 1634) | 40.1 % (222 of 553) | 66.8 % (545 of 816) | 73.6 % (195 of 265) |
Sidechain | 15.1 % (301 of 1998) | 9.1 % (109 of 1204) | 25.0 % (192 of 768) | 0.0 % (0 of 26) |
Aromatic | 0.0 % (0 of 238) | 0.0 % (0 of 119) | 0.0 % (0 of 119) | |
Methyl | 17.5 % (62 of 354) | 14.7 % (26 of 177) | 20.3 % (36 of 177) |
1. PPARgamma LBD
GQLNPESADL RALAKHLYDS YIKSFPLTKA KARAILTGKT TDKSPFVIYD MNSLMMGEDK IKFKHITPLQ EQSKEVAIRI FQGCQFRSVE AVQEITEYAK SIPGFVNLDL NDQVTLLKYG VHEIIYTMLA SLMNKDGVLI SEGQGFMTRE FLKSLRKPFG DFMEPKFEFA VKFNALELDD SDLAIFIAVI ILSGDRPGLL NVKPIEDIQD NLLQALELQL KLNHPESSQL FAKLLQKMTD LRQIVTEHVQ LLQVIKKTET DMSLHPLLQE IYKDLYSolvent system 90% H2O/10% D2O, Pressure 1 atm, Temperature 298 K, pH 7.4
# | Name | Isotope labeling | Type | Concentration |
---|---|---|---|---|
1 | PPARgamma LBD | [U-100% 13C; U-100% 15N; U-80% 2H] | 1 mM | |
2 | MRL24 | natural abundance | 1 mM |